Activity of piperaquine and other 4-aminoquinoline antiplasmodial drugs against chloroquine-sensitive and resistant blood-stages of Plasmodium falciparum. Role of β-haematin inhibition and drug concentration in vacuolar water- and lipid-phases

  • David C. Warhurst
  • , John C. Craig
  • , Ipemida S. Adagu
  • , R. Kiplin Guy
  • , Peter B. Madrid
  • , Quinton L. Fivelman

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85 Scopus citations

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Pharmacology, Toxicology and Pharmaceutical Science