Chemistry of insect antifeedants from Azadirachta indica (Part 20): Synthesis of biologically active, simple analogues of azadirachtin, containing the hydroxytetrahydrofurancarboxylate hemiketal moiety

María L. De La Puente; Robert B. Grossman; Steven V. Ley; Monique S.J. Simmonds; Wally M. Blaney

doi:10.1039/p19960001517

Chemistry of insect antifeedants from Azadirachta indica (Part 20): Synthesis of biologically active, simple analogues of azadirachtin, containing the hydroxytetrahydrofurancarboxylate hemiketal moiety

María L. De La Puente, Robert B. Grossman, Steven V. Ley, Monique S.J. Simmonds, Wally M. Blaney

Chemistry

Research output: Contribution to journal › Article › peer-review

9 Scopus citations

Abstract

A synthetic route to mimics of the insect antifeedant azadirachtin 1 containing the hydroxytetrahydrofurancarboxylate hemiketal functional moiety has been developed. Two of these compounds, 2 and 11, show significant antifeedant activity against Spodoptera littoralis, although they are not as active as azadirachtin.

Original language	English
Pages (from-to)	1517-1521
Number of pages	5
Journal	Journal of the Chemical Society - Perkin Transactions 1
Issue number	13
DOIs	https://doi.org/10.1039/p19960001517
State	Published - Jul 7 1996

ASJC Scopus subject areas

General Chemistry

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10.1039/p19960001517

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De La Puente, M. L., Grossman, R. B., Ley, S. V., Simmonds, M. S. J., & Blaney, W. M. (1996). Chemistry of insect antifeedants from Azadirachta indica (Part 20): Synthesis of biologically active, simple analogues of azadirachtin, containing the hydroxytetrahydrofurancarboxylate hemiketal moiety. Journal of the Chemical Society - Perkin Transactions 1, (13), 1517-1521. https://doi.org/10.1039/p19960001517

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abstract = "A synthetic route to mimics of the insect antifeedant azadirachtin 1 containing the hydroxytetrahydrofurancarboxylate hemiketal functional moiety has been developed. Two of these compounds, 2 and 11, show significant antifeedant activity against Spodoptera littoralis, although they are not as active as azadirachtin.",

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De La Puente, ML, Grossman, RB, Ley, SV, Simmonds, MSJ & Blaney, WM 1996, 'Chemistry of insect antifeedants from Azadirachta indica (Part 20): Synthesis of biologically active, simple analogues of azadirachtin, containing the hydroxytetrahydrofurancarboxylate hemiketal moiety', Journal of the Chemical Society - Perkin Transactions 1, no. 13, pp. 1517-1521. https://doi.org/10.1039/p19960001517

Chemistry of insect antifeedants from Azadirachta indica (Part 20): Synthesis of biologically active, simple analogues of azadirachtin, containing the hydroxytetrahydrofurancarboxylate hemiketal moiety. / De La Puente, María L.; Grossman, Robert B.; Ley, Steven V. et al.
In: Journal of the Chemical Society - Perkin Transactions 1, No. 13, 07.07.1996, p. 1517-1521.

Research output: Contribution to journal › Article › peer-review

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De La Puente ML, Grossman RB, Ley SV, Simmonds MSJ, Blaney WM. Chemistry of insect antifeedants from Azadirachta indica (Part 20): Synthesis of biologically active, simple analogues of azadirachtin, containing the hydroxytetrahydrofurancarboxylate hemiketal moiety. Journal of the Chemical Society - Perkin Transactions 1. 1996 Jul 7;(13):1517-1521. doi: 10.1039/p19960001517

Chemistry of insect antifeedants from Azadirachta indica (Part 20): Synthesis of biologically active, simple analogues of azadirachtin, containing the hydroxytetrahydrofurancarboxylate hemiketal moiety

Abstract

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