Identification and characterization of inhibitors of the aminoglycoside resistance acetyltransferase Eis from Mycobacterium tuberculosis

Keith D. Green, Wenjing Chen, Sylvie Garneau-Tsodikova

Research output: Contribution to journalArticlepeer-review

59 Scopus citations
Original languageEnglish
Pages (from-to)73-77
Number of pages5
JournalChemMedChem
Volume7
Issue number1
DOIs
StatePublished - Jan 2 2012

Keywords

  • Aminoglycoside acetyltransferase
  • Antibiotics
  • Bacterial resistance
  • Eis protein
  • High-throughput screening
  • Inhibitors

ASJC Scopus subject areas

  • Drug Discovery
  • General Pharmacology, Toxicology and Pharmaceutics
  • Molecular Medicine
  • Biochemistry
  • Pharmacology
  • Organic Chemistry

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